Search results for "Cholesterol side-chain cleavage enzyme"

showing 3 items of 3 documents

Neurosteroidogenesis in Rat Retinas

2002

Neurosteroids (steroids synthesized in the CNS) function by modulating neurotransmission. To establish an experimental model for investigation of neurosteroid synthesis and regulation, independent of blood-borne steroids, we examined the steroidogenic activity of isolated rat retinas. We identified progesterone, pregnenolone, dehydroepiandrosterone, desoxycorticosterone, 3 alpha,5 alpha-tetrahydrodesoxycorticosterone, 3 alpha-hydroxy-5 alpha-dihydroprogesterone, 17-hydroxyprogesterone, and 17-hydroxypregnenolone together with their esterified forms. As pregnenolone is the precursor of all steroids, its formation was studied in detail as an index of a steroid-synthesizing tissue. Pregnenolon…

Central Nervous SystemMaleTime FactorsNeuroactive steroidDehydroepiandrosteroneBiochemistryGas Chromatography-Mass SpectrometryRetinaCellular and Molecular NeuroscienceCyclic AMPmedicineAnimalsCholesterol Side-Chain Cleavage EnzymeLovastatinRats WistarChromatography High Pressure LiquidProgesteroneNeurotransmitter AgentsDose-Response Relationship DrugbiologyCholesterol side-chain cleavage enzymeCytochrome P450DehydroepiandrosteroneAminoglutethimideImmunohistochemistryRatsmedicine.anatomical_structureBiochemistryPregnenoloneInner nuclear layerPregnenolonebiology.proteinSteroidsLovastatinAminoglutethimidemedicine.drugJournal of Neurochemistry
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Human neuroblastoma SH-SY5Y cell line: neurosteroid-producing cell line relying on cytoskeletal organization.

2000

Pregnenolone, the precursor of all steroids, is synthesized by CNS structures. The synthesis requires an obligatory step involving cholesterol transport to mitochondrial cytochrome P450-cholesterol side chain cleavage (cytP450scc), although the underlying mechanism(s) are still mostly unknown. We used the human neuroblastoma SH-SY5Y cell line to investigate cytP450scc expression and activity and to establish a role of cytoskeleton in pregnenolone synthesis. Immunocytochemical and biochemical approaches revealed that undifferentiated as well as differentiated cells either by retinoic acid (RA) or phorbol ester 12-O-tetradecanoylphorbol-13-acetate (TPA), possess cytP450scc and rapidly synthes…

Central Nervous SystemSH-SY5YNeuroactive steroidCellular differentiationRetinoic acidTrilostaneBiologyCellular and Molecular Neurosciencechemistry.chemical_compoundNeuroblastomachemistryBiochemistryCytochrome P-450 Enzyme SystemCell culturePregnenolonemedicinePregnenoloneTumor Cells CulturedHumansSteroidsCholesterol Side-Chain Cleavage EnzymeCytoskeletonCytoskeletonmedicine.drugJournal of neuroscience research
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Biosynthesis and transformation of 20α 21-dihydroxycholesterol by rat adrenal preparations

1979

Abstract The biosynthesis of [ 3 H]-20α, 21 dihydroxycholestderol from [ 3 H]-20α-hydroxycholesterol and its transformation to [ 3 H]-21-hydroxypregnenolone by rat adrenal preparations has been demonstrated. 20α-Hydroxycholesterol was transformed to 20α, 21-dihydroxycholesterol by microsomal preparations in the presence of NADPH and 20α-21-dihydroxycholesterol was metabolized to 21-hydroxypregnenolone by mitochondrial preparations in the presence of a NADPH-generating-system. Comparison of the Michaelis-Menten-Kinetics of the steps “20α, 21-dihydroxycholesterol → 21-hydroxycholesterol” and “20α-hydroxycholesterol → pregnenolone” revealed that both compounds behaved as analogue substrates of…

Malemedicine.drug_classStereochemistryBiology17-alpha-HydroxypregnenoloneBiochemistrychemistry.chemical_compoundEndocrinologyBiosynthesisMicrosomesAdrenal Glandspolycyclic compoundsmedicineAnimalsCholesterol Side-Chain Cleavage EnzymeCholesterol side-chain cleavage enzymeHydroxycholesterolsMitochondriaRatsTransformation (genetics)BiochemistrychemistryAlternative complement pathwayPregnenoloneMicrosomeCorticosteroidlipids (amino acids peptides and proteins)NADPmedicine.drugJournal of Steroid Biochemistry
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